The search for new COX-2 inhibitors: a review of 2002 - 2008 patents

Registro completo de metadados
MetadadosDescriçãoIdioma
Autor(es): dc.creatorRamalho, Teodorico C.-
Autor(es): dc.creatorRocha, Marcus V. J.-
Autor(es): dc.creatorCunha, Elaine F. F. da-
Data de aceite: dc.date.accessioned2026-02-09T12:31:42Z-
Data de disponibilização: dc.date.available2026-02-09T12:31:42Z-
Data de envio: dc.date.issued2017-10-11-
Data de envio: dc.date.issued2017-10-11-
Data de envio: dc.date.issued2009-
Fonte completa do material: dc.identifierhttps://repositorio.ufla.br/handle/1/15528-
Fonte completa do material: dc.identifierhttp://www.tandfonline.com/doi/abs/10.1517/13543770903059125?journalCode=ietp20-
Fonte: dc.identifier.urihttp://educapes.capes.gov.br/handle/capes/1163099-
Descrição: dc.descriptionBackground: Two COX isoenzymes are known, COX-1 and COX-2, for which the main inhibitors are the NSAIDs. The common anti-inflammatory drugs (such as aspirin, ibuprofen and naproxen) all act by blocking the action of both the COX-1 and COX-2 enzymes. The COX-2 inhibitors represent a new class of drugs that do not affect COX-1 but selectively block COX-2. This selective action provides the benefits of reducing inflammation without irritating the stomach and cardiovascular effects. Objective: This review focuses on patents published in the field during 2002 – 2008, paying particular attention to promising COX-2 inhibitors. Conclusion: Structural analogues of the COX-2 inhibitors celecoxib and valdecoxib, and novel potential pyridazine, triazole, indole and thione derivatives emerge as promising leads for the treatment of inflammation, pain and other diseases.-
Idioma: dc.languageen-
Publicador: dc.publisherTaylor & Francis-
Direitos: dc.rightsrestrictAccess-
???dc.source???: dc.sourceExpert Opinion on Therapeutic Patents-
Palavras-chave: dc.subjectAnti-inflammatory drugs-
Palavras-chave: dc.subjectCOX-2-
Palavras-chave: dc.subjectNSAIDs-
Palavras-chave: dc.subjectAnti-inflamatórios-
Título: dc.titleThe search for new COX-2 inhibitors: a review of 2002 - 2008 patents-
Tipo de arquivo: dc.typeArtigo-
Aparece nas coleções:Repositório Institucional da Universidade Federal de Lavras (RIUFLA)

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