The Challenges of Antitubercular Drug Discovery

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MetadadosDescriçãoIdioma
Autor(es): dc.contributorUniversidade Estadual Paulista (UNESP)-
Autor(es): dc.contributorUnidad de Posgrado en Farmacia y Bioquímica-
Autor(es): dc.creatorPrates, João Lucas Bruno-
Autor(es): dc.creatordos Santos Fernandes, Guilherme Felipe-
Autor(es): dc.creatorRodríguez-Silva, Cristhian N.-
Autor(es): dc.creatordos Santos, Jean Leandro-
Data de aceite: dc.date.accessioned2025-08-21T17:48:46Z-
Data de disponibilização: dc.date.available2025-08-21T17:48:46Z-
Data de envio: dc.date.issued2025-04-29-
Data de envio: dc.date.issued2022-12-31-
Fonte completa do material: dc.identifierhttp://dx.doi.org/10.1007/978-3-031-15955-8_23-
Fonte completa do material: dc.identifierhttps://hdl.handle.net/11449/298445-
Fonte: dc.identifier.urihttp://educapes.capes.gov.br/handle/11449/298445-
Descrição: dc.descriptionAlthough extensive efforts have been undertaken to eradicate tuberculosis (TB), it remains one of the deadliest infections. The rising number of drug-resistant strainsStraindrug-resistant contributing to high mortalityMortality rates has become a global concern, highlighting the need for suitable treatments to eliminate such strains. However, the limitations of current therapies are long treatment duration, adverse side effectsSide effect, interactions with other drugs, toxicity, and poor efficacyEfficacy against latent strains. Thus, the search for safe and effective anti-TB drugsDruganti-TB is urgent. This chapter addresses the advances and challengesChallenge in drug discoveryDiscoverydrug for treating TB by focusing on the recently approved drugsDrugApproved and the most promising candidatesCandidate that can contribute to current therapies. Antitubercular drug discovery: challenges-
Descrição: dc.descriptionSão Paulo State University (UNESP) Institute of Chemistry-
Descrição: dc.descriptionUniversidad Nacional de Trujillo Escuela de Posgrado Unidad de Posgrado en Farmacia y Bioquímica-
Descrição: dc.descriptionSchool of Pharmaceutical Sciences São Paulo State University (UNESP), Rodovia Araraquara-Jaú Km 1, S/N, Campus Ville-
Descrição: dc.descriptionSão Paulo State University (UNESP) Institute of Chemistry-
Descrição: dc.descriptionSchool of Pharmaceutical Sciences São Paulo State University (UNESP), Rodovia Araraquara-Jaú Km 1, S/N, Campus Ville-
Formato: dc.format483-498-
Idioma: dc.languageen-
Relação: dc.relationIntegrated Science-
???dc.source???: dc.sourceScopus-
Palavras-chave: dc.subjectAntitubercular drugs-
Palavras-chave: dc.subjectDrug design-
Palavras-chave: dc.subjectMycobacterium tuberculosis-
Palavras-chave: dc.subjectNew drugs-
Palavras-chave: dc.subjectTuberculosis-
Título: dc.titleThe Challenges of Antitubercular Drug Discovery-
Tipo de arquivo: dc.typelivro digital-
Aparece nas coleções:Repositório Institucional - Unesp

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