Recent Trends in Drug Development for the Treatment of Adenocarcinoma Breast Cancer: Thiazole, Triazole, and Thiosemicarbazone Analogues as Efficient Scaffolds

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MetadadosDescriçãoIdioma
Autor(es): dc.contributorUniversidade Estadual Paulista (UNESP)-
Autor(es): dc.contributorLapdesf-Laboratory of Research and Development of Drugs-
Autor(es): dc.contributorUnion of the Colleges of the Great Lakes (UNILAGO)-
Autor(es): dc.creatorScarim, Cauê Benito-
Autor(es): dc.creatorChin, Chung Man-
Data de aceite: dc.date.accessioned2025-08-21T19:30:01Z-
Data de disponibilização: dc.date.available2025-08-21T19:30:01Z-
Data de envio: dc.date.issued2023-03-02-
Data de envio: dc.date.issued2023-03-02-
Data de envio: dc.date.issued2022-07-01-
Fonte completa do material: dc.identifierhttp://dx.doi.org/10.2174/1871520621666211201152815-
Fonte completa do material: dc.identifierhttp://hdl.handle.net/11449/241875-
Fonte: dc.identifier.urihttp://educapes.capes.gov.br/handle/11449/241875-
Descrição: dc.descriptionThiazoles, triazoles, and thiosemicarbazones function as efficient scaffolds in compounds for the treatment of several illnesses, including cancers. In this review article, we have demonstrated various studies involving these three pharmacophore classes (thiazoles, triazoles, and thiosemicarbazones) in medicinal chemistry over the last decade (2011-2021) with a focus on MCF-7 adenocarcinoma breast cancer cells. Our objective is to facilitate drug discovery of novel chemotherapeutic agents by detailing anti-proliferative compounds.-
Descrição: dc.descriptionCoordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES)-
Descrição: dc.descriptionFundação de Amparo à Pesquisa do Estado de São Paulo (FAPESP)-
Descrição: dc.descriptionSchool of Pharmaceutical Sciences Sao Paulo State University (UNESP), SP-
Descrição: dc.descriptionLapdesf-Laboratory of Research and Development of Drugs, SP-
Descrição: dc.descriptionAdvanced Research Center in Medicine (CEPAM) School of Medicine Union of the Colleges of the Great Lakes (UNILAGO), SP-
Descrição: dc.descriptionSchool of Pharmaceutical Sciences Sao Paulo State University (UNESP), SP-
Descrição: dc.descriptionCAPES: 001-
Descrição: dc.descriptionFAPESP: 2016/10847-9-
Formato: dc.format2204-2240-
Idioma: dc.languageen-
Relação: dc.relationAnti-Cancer Agents in Medicinal Chemistry-
???dc.source???: dc.sourceScopus-
Palavras-chave: dc.subjectanti-proliferative-
Palavras-chave: dc.subjectbreast cancer-
Palavras-chave: dc.subjectMCF-7-
Palavras-chave: dc.subjectThiazoles-
Palavras-chave: dc.subjectthiosemicarbazones-
Palavras-chave: dc.subjecttriazoles-
Título: dc.titleRecent Trends in Drug Development for the Treatment of Adenocarcinoma Breast Cancer: Thiazole, Triazole, and Thiosemicarbazone Analogues as Efficient Scaffolds-
Tipo de arquivo: dc.typevídeo-
Aparece nas coleções:Repositório Institucional - Unesp

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