Insight into Recent Drug Discoveries against Trypanosomatids and Plasmodium spp Parasites: New Metal-based Compounds

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MetadadosDescriçãoIdioma
Autor(es): dc.contributorUniversidade Estadual Paulista (UNESP)-
Autor(es): dc.contributorUnion of the Colleges of the Great Lakes (UNILAGO)-
Autor(es): dc.creatorScarim, Cauê Benito-
Autor(es): dc.creatorde Farias, Renan Lira-
Autor(es): dc.creatorChiba, Diego Eidy-
Autor(es): dc.creatorChin, Chung Man-
Data de aceite: dc.date.accessioned2025-08-21T17:24:45Z-
Data de disponibilização: dc.date.available2025-08-21T17:24:45Z-
Data de envio: dc.date.issued2023-03-02-
Data de envio: dc.date.issued2023-03-02-
Data de envio: dc.date.issued2022-04-01-
Fonte completa do material: dc.identifierhttp://dx.doi.org/10.2174/0929867328666210917114912-
Fonte completa do material: dc.identifierhttp://hdl.handle.net/11449/241818-
Fonte: dc.identifier.urihttp://educapes.capes.gov.br/handle/11449/241818-
Descrição: dc.descriptionScaffolds of metal-based compounds can act as pharmacophore groups in several ligands to treat various diseases, including tropical infectious diseases (TID). In this review article, we investigate the contribution of these moieties to medicinal inorganic chemistry in the last seven years against TID, including American trypanosomiasis (Chagas disease), human African trypanosomiasis (HAT, sleeping sickness), leishmania, and malaria. The most potent metal-based complexes are displayed and highlighted in figures, tables and graphics; according to their pharmacological activities (IC50 > 10µM) against Trypanosomatids and Plasmodium spp parasites. We highlight the current progresses and viewpoints of these metal-based complexes, with a specific focus on drug discovery.-
Descrição: dc.descriptionCoordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES)-
Descrição: dc.descriptionFundação de Amparo à Pesquisa do Estado de São Paulo (FAPESP)-
Descrição: dc.descriptionSao Paulo State University(UNESP) School of Pharmaceutical Sciences, SP-
Descrição: dc.descriptionLapdesf-Laboratory of Research and Development of Drugs Sao Paulo State University (UNESP) School of Pharmaceutical Sciences, SP-
Descrição: dc.descriptionSao Paulo State University(UNESP) Institute of Chemistry, SP-
Descrição: dc.descriptionAdvance Research Center in Medicine Union of the Colleges of the Great Lakes (UNILAGO), SP-
Descrição: dc.descriptionSao Paulo State University(UNESP) School of Pharmaceutical Sciences, SP-
Descrição: dc.descriptionLapdesf-Laboratory of Research and Development of Drugs Sao Paulo State University (UNESP) School of Pharmaceutical Sciences, SP-
Descrição: dc.descriptionSao Paulo State University(UNESP) Institute of Chemistry, SP-
Descrição: dc.descriptionCAPES: 001-
Descrição: dc.descriptionFAPESP: 2016/10847-9-
Formato: dc.format2334-2381-
Idioma: dc.languageen-
Relação: dc.relationCurrent Medicinal Chemistry-
???dc.source???: dc.sourceScopus-
Palavras-chave: dc.subjectLeishmania-
Palavras-chave: dc.subjectMetal-based drugs-
Palavras-chave: dc.subjectnew drugs-
Palavras-chave: dc.subjectPlasmodium ssp-
Palavras-chave: dc.subjectT. brucei-
Palavras-chave: dc.subjectT. cruzi-
Título: dc.titleInsight into Recent Drug Discoveries against Trypanosomatids and Plasmodium spp Parasites: New Metal-based Compounds-
Tipo de arquivo: dc.typevídeo-
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